News

Unibest NewCo & Licensing Pipeline

Views: 1778     Author: Unibest Industrial     Publish Time: 2025-12-01      Origin: Site

facebook sharing button
twitter sharing button
line sharing button
wechat sharing button
linkedin sharing button
pinterest sharing button
sharethis sharing button

Last Updated: 2025-12-01

Antibody-Drug Conjugate (ADC)

CodeTargetIndicationPreclinicalPh IPh IIPh IIINDA/BLADetail
UB410HER2Metastatic breast cancer

UB409HER2HER2-positive breast cancer

UB391Her2/Her2Breast cancer; Esophageal cancer; Gastric cancer; Non-small cell lung cancer

UB390ROR1Solid tumour; Haematologic malignancy

UB044Microtubule (ADC payload)HER2-negative breast cancer; HER2-positive gastric cancer

UB320ROR1; DNA Topoisomerase IDiffuse large B-cell lymphoma

UB322MUC17; DNA Topoisomerase ISolid tumour

UB323FGFR2b; DNA Topoisomerase ISolid tumour

UB319ROR1; DNA Topoisomerase ISolid tumour

UB318ROR1; DNA Topoisomerase IMantle cell lymphoma; Diffuse large B-cell lymphoma; Classical Hodgkin's disease

UB424BCMAMultiple myeloma

UB321CDH17; DNA Topoisomerase IGastrointestinal cancer

UB394GPC3Solid tumour

UB392CLDN6Solid tumour

UB393ITGB6Solid tumour

UB022HER2/Trop2Breast cancer; Cervical cancer; Gastric cancer

UB032Nectin-4/Trop2Bladder cancer; Cervical cancer; Lung cancer

UB031cMet/HER2Pancreatic cancer; Lung cancer; Gastrointestinal cancer; Renal cancer

UB127EGFR; cMetLung cancer

UB126ADAM9Gastrointestinal cancer

UB191TROP2 BsAb + Dual-payloadPancreatic cancer

UB138Undisclosed (BsAb+Dual-payload)Solid tumour

UB137Undisclosed (mAb+Dual-payload)Solid tumour

UB136BsAb + Dual-payloadSolid tumour

UB431DLL3 BsAb + Dual-payloadSmall cell lung cancer; Neuroendocrine tumour

UB189B7H3 BsAb + Dual-payloadSmall cell lung cancer

UB190B7H3 Bi-functional+ Dual-payloadProstate cancer

Antibody

CodeTargetIndicationPreclinicalPh IPh IIPh IIINDA/BLADetail
UB493
Non-small cell lung cancer; Colorectal cancer metastatic

UB186EGFRColorectal cancer
About
UB187PD1Recurrent thymic carcinoma; Metastatic thymic carcinoma

UB302VEGF-ANeovascular age-related macular degeneration

UB335IL-6RRheumatoid arthritis

UB336IL-6RIdiopathic multicentric Castleman disease

UB331IL-4RαAtopic dermatitis
About
UB330IL-4RαPrurigo nodularis
About
UB426IL4Atopic dermatitis; Prurigo nodularis; Asthma

UB396EGFR/cMetSolid tumour

UB014EGFR; CD3Breast cancer metastatic; Gastric cancer
About
UB408BCMA/CD3Multiple myeloma; Primary amyloidosis

UB013LAG3Solid tumour; Lymphoma; Autoimmune disorder
About
UB017IL-12 prodrugSolid tumour
About
UB149AβAlzheimer's disease

UB385IL36RAutoimmune disorder

UB423PDL1 x VEGF x TGFbSolid tumour

UB015EGFR; CD3 (enzyme-controlled)Solid tumour
About
UB019GPC3; CD3Hepatocellular carcinoma
About
UB427OX40L x TNFα; OX40LAtopic dermatitis; Hidradenitis suppurativa; Asthma

UB333(BsAb)IgA nephropathy

UB332(BsAb)Inflammatory bowel disease; Psoriasis; Psoriatic arthritis

UB266CD38Multiple myeloma (MM); Multiple myeloma

UB340TL1AInflammatory bowel disease; Ulcerative colitis; Crohn's disease; Systemic sclerosis

UB343TL1A; IL-6RInflammatory bowel disease; Thyroid eye disease

UB341TL1A; IL-23p19Inflammatory bowel disease; Psoriasis

UB342TL1A; TNF-αInflammatory bowel disease; Rheumatoid arthritis

UB345IL-6R; TNF-αUveitis; Neuromyelitis optica spectrum disorder; Dental caries

UB344IL-6R; IL-23p19Rheumatoid arthritis; Thyroid eye disease; Chronic kidney disease; Atherosclerotic cardiovascular disease

UB267CD38Multiple myeloma

UB018RORI; CD3Lymphoma; Breast cancer

UB023PD-L1; VEGFLung cancer; Breast cancer

UB041HERV-K Env-TMMalignant neoplasm

UB020PD-1/IL-15 cytokine antibody conjudgateSolid tumour
About
UB377ActRIIA/BObesity

Cell and Gene Therapy (CGT)

CodeTargetIndicationPreclinicalPh IPh IIPh IIINDA/BLADetail
UB425CD19Diffuse large B-cell lymphoma; Mantle cell lymphoma; Acute lymphoblastic leukaemia

UB098HBVHepatocellular carcinoma
About
UB038TGFβ1; COX-2 (siRNA)Non-melanoma skin cancer
About
UB084(Oncolytic virus)Head and neck squamous cell carcinoma; Lung cancer; Ovarian cancer; Sarcoma; Triple negative breast cancer
About
UB039TGFβ1; COX-2 (siRNA)Localised adiposity
About
UB145Factor XI (siRNA)Anticoagulant therapy; Stroke

UB144(siRNA)Solid tumour

UB139PCSK9 (siRNA)Hypercholesterolaemia

UB354
Varicella zoster virus infection

UB099HBVCholangiocarcinoma
About
UB499
Malignant neoplasm

UB494CD7T-cell acute lymphoblastic leukaemia; Lymphoblastic lymphoma

UB496
Neoplasm malignant

UB140PCSK9 (siRNA)Hypercholesterolaemia

UB101HPVCervical cancer; Head and neck cancer
About
UB100HBVChronic hepatitis B
About
UB085(Oncolytic virus)Head and neck squamous cell carcinoma; Lung cancer; Ovarian cancer; Sarcoma; Triple negative breast cancer
About
UB495
Neoplasm malignant

UB355
Tuberculosis

UB356
Malignant neoplasm

UB095(siRNA)Nephrotic syndrome

UB089IL4R (siRNA)Atopic dermatitis

UB092(siRNA)Age-related macular degeneration

UB090Calcineurin/Fn14 (siRNA)Transplantation; Autoimmune disorder

UB146ApoC3 (siRNA)Hypertriglyceridaemia

UB498
Malignant neoplasm; Infection

UB097(siRNA)Melanoma

UB102EBVSolid tumour
About
UB096SGLT2 (siRNA)Type 2 diabetes mellitus; Gout

UB103(iPSC)Solid tumour
About
UB418RetinaRetinal degeneration

UB091Glucosylceramide synthase (siRNA)Gaucher's disease; Fabry's disease

UB093Renin / AGTHypertension

UB094FcRn (siRNA)Myasthenia gravis

Fusion Protein

CodeTargetIndicationPreclinicalPh IPh IIPh IIINDA/BLADetail
UB350GLP-1; GLP-2Obesity; Type 2 diabetes mellitus

UB325FGF21R; GCGR; GLP-1 RMetabolic dysfunction-associated fatty liver disease
About
UB326FGF21R; GCGR; GLP-1 RHypertriglyceridaemia
About
UB421GLP-1 x GCG x FGF21Metabolic dysfunction-associated steatohepatitis; Symptomatic Human Thyroidal Group

UB337CD80; CD86Rheumatoid arthritis; Systemic lupus erythematosus; Graft versus host disease

UB329CLDN18.2Solid tumour
About
UB328PDL1; VEGF; TGFβGastrointestinal cancer
About
UB327PDL1; VEGF; TGFβNon-small cell lung cancer
About
UB338IL-1R1Cryopyrin-associated periodic syndromes; Gouty arthritis

UB352αActRII; αMyostatinObesity

UB351GLP-1; GLP-2Obesity

Peptide

CodeTargetIndicationPreclinicalPh IPh IIPh IIINDA/BLADetail
UB011GLP-1 RDiabetes mellitus
About
UB430Insulin receptorDiabetes

UB080GLP-1Obesity
About
UB298Insulin receptorType 2 diabetes mellitus

UB045GLP-1Type 2 diabetes mellitus
About
UB081GLP-1Nonalcoholic steatohepatitis
About
UB316GLP-1; GIPDiabetes mellitus

UB315GLP-1; GIPObesity; Overweight

UB012GLP-1 RObesity
About
UB411Functional fragment of Thymosin β4Corneal epithelial defect; Pterygium; Neurotrophic keratitis

UB047GLP-1; GCGObesity
About
UB285Tumor neuantigensPancreatic cancer
About
UB048GLP-1; GCGNonalcoholic steatohepatitis
About
UB049ÎĽ opioid receptorOpioid-induced constipation
About
UB317GLP-1; GIPNonalcoholic fatty liver disease; Nonalcoholic steatohepatitis; Obstructive sleep apnoea syndrome; Cardiac failure with preserved ejection fraction

UB046GLP-1Type 2 diabetes mellitus
About
UB050GCGRCongenital hyperinsulinism
About
UB263GLP-1 RType 2 diabetes mellitus
About
UB051GLP-1; GIPType 2 diabetes mellitus; Obesity; Nonalcoholic steatohepatitis
About
UB052GLP-1R; GIPR; GCGRType 2 diabetes mellitus; Obesity; Metabolic dysfunction-associated steatohepatitis
About
UB104GLP-1 (Oromucosal)Diabetes mellitus; Obesity

UB010GLP-1 RDiabetes mellitus
About

Polysaccharide

CodeTargetIndicationPreclinicalPh IPh IIPh IIINDA/BLADetail
UB432TLR9Peritoneal carcinomatosis; Solid tumour

Protein

CodeTargetIndicationPreclinicalPh IPh IIPh IIINDA/BLADetail
UB434
Ischaemic stroke

UB433
Amyotrophic lateral sclerosis

UB437
Multiple system atrophy; CADASIL

UB436
Traumatic brain injury

UB435
Alzheimer's disease

UB438
Amyotrophic lateral sclerosis

UB412
Diabetic macular oedema; Exudative age-related macular degeneration

UB439
Autism spectrum disorder

Biologics

CodeTargetIndicationPreclinicalPh IPh IIPh IIINDA/BLADetail
UB339TregInflammatory bowel disease; Amyotrophic lateral sclerosis; Systemic lupus erythematosus

Small Molecule

CodeTargetIndicationPreclinicalPh IPh IIPh IIINDA/BLADetail
UB202Lanosterol 14-alpha demethylaseInvasive aspergillosis; Mucormycosis
ANDA

UB422NeuroprotectiveCerebrovascular accident

UB082F protein (RSV)Respiratory syncytial virus infection
About
UB360P2Y12RPeripheral arterial disease
About
UB395CDK2/4/6Breast cancer metastatic; Liposarcoma; Lung cancer metastatic

UB314EGFR (L858R)Non-small cell lung cancer

UB068JAK1 (oral)Ankylosing spondylitis
About
UB312GLP-1 (oral)Obesity; Overweight

UB309JAK1; JAK2Vitiligo

UB313GLP-1 (oral)Diabetes mellitus

UB384PDE3/4Chronic obstructive pulmonary disease

UB353SYK inhibitorImmune thrombocytopenia

UB361JAK1 (oral)Atopic dermatitis
About
UB063HBV CaspidChronic hepatitis B
About
UB428PDE4Psoriasis; Atopic dermatitis

UB429Steroid + VDPsoriasis

UB062KCNQ2/3Epilepsy
About
UB347Core Protein CpAMHepatitis B

UB348Surface Antigen HBsAgHepatitis B

UB386AT2RPost-stroke pain

UB310JAK1; JAK2Prurigo nodularis

UB362JAK1 (oral)Vitiligo
About
UB067JAK1 (Gel)Atopic dermatitis
About
UB0425-HT; DAAutism spectrum disorder; Atrial septal defect; Acute stress disorder
About
UB024KV1.3 (Topical)Atopic dermatitis
About
UB027mTORC2Neuroendocrine tumour; Lung cancer; Breast cancer

UB064TEADMalignant neoplasm
About
UB387BTKHaematological malignancy

UB397EGFRLung cancer

UB388ARMetastatic castration-resistant prostate cancer

UB364JAK1 (oral)Rheumatoid arthritis
About
UB028FXIaThrombus

UB026PI3K-Akt-mTOR pathwayMalignant melanoma; Oesophageal cancer; Colorectal cancer

UB176KV1.3 (Topical)Psoriasis
About
UB147Keratin; Plasmin

UB083F protein (RSV)Respiratory syncytial virus infection prophylaxis
About
UB349ASK-1Nonalcoholic steatohepatitis; Hepatic fibrosis

UB363JAK1 (oral)Inflammatory bowel disease
About
UB069RIPK1Peripheral arterial disease; Primary biliary cholangitis
About
UB497
Cervical intraepithelial neoplasia

UB509IDH1 mutationLow grade glioma; Cholangiocarcinoma; Chondrosarcoma

UB365TRKA (Gel)Skin inflammation; Pruritus
About
UB148Androgen receptor

UB029KV1.3 (Oral)Inflammatory bowel disease
About
UB030cMyc pathwayGynaecological neoplasm

UB177KV1.3 (Oral)Atopic dermatitis
About
UB284AChEMyasthenia gravis

UB404MENINHaematological malignancy

UB398Pan KRASSolid tumour

UB376GLP-1RObesity

UB366TRKA/B/CSolid tumour
About
UB389ERBreast cancer

UB401USP1Solid tumour

UB400PARP1Solid tumour; Brain metastases

UB125GABAA ReceptorEpilepsy

UB183Ion channel inhibitorDiabetic nephropathy
About
UB178KV1.3 (Topical)Alopecia
About
UB179GPCRDiabetic retinopathy; Age-related macular degeneration
About
UB065P2Y12RAcute coronary syndrome
About
UB066P2Y12RIschaemic stroke
About
UB070pan-RAS (on)Solid tumour
About
UB043Agmatinase; Imidazoline Rc; NMDA RcAtrial septal defect; Autism spectrum disorder; Acute stress disorder
About
UB040Multiple targets; immunostimulantsMalignant neoplasm

UB182Ion channel inhibitorPruritus
About
UB180GPCROcular inflammation
About
UB181GPCRChronic obstructive pulmonary disease
About
UB413
Retinoblastoma

UB367IL-17Psoriasis

UB369ER-PROTACBreast cancer

UB368BTK-PROTACSystemic lupus erythematosus; Atopic dermatitis

UB371MAT2ASolid tumour

UB370ATMSolid tumour

UB372WRNSolid tumour

UB380GIPRDiabetes mellitus

UB381STAT6Autoimmune disorder; Respiratory disorder

UB373
Inflammatory bowel disease

UB375
Weight decreased

UB374
Diabetes mellitus; Obesity

UB399Pan RASSolid tumour

UB406KEAP1Solid tumour

UB402PRMT5Solid tumour

UB407WFS1Solid tumour

UB405BTKChronic lymphocytic leukaemia; Small lymphocytic lymphoma; Diffuse large B-cell lymphoma

UB403POLQSolid tumour

UB383VAV1Autoimmune disorder

UB382NEK7-MGDAutoimmune disorder

UB378ActRIIBObesity

UB379AMYRObesity; Diabetes mellitus

Targeted Protein Degradation

CodeTargetIndicationPreclinicalPh IPh IIPh IIINDA/BLADetail
UB025cMycPancreatic cancer

UB324HPK-1Solid tumour